Pharmacokinetic parameters | FCTa PO 2 mg/kg | ODFb PO 2 mg/kg | Rectalc 2 mg/kg | Rectal 10 mg/kg |
---|---|---|---|---|
Cmax (μg/mL) | 0.21 ± 0.07 | 0.25 ± 0.10 | 0.09 ± 0.04 | 0.26 ± 0.08 |
Tmax (hours) | 2.08 ± 1.30 | 1.88 ± 1.65 | 3.28 ± 2.49 | 4.30 ± 2.91 |
T1/2 (hours) | 5.46 ± 2.39 | 4.62 ± 1.49 | 4.82 ± 1.91 | 4.20 ± 1.40 |
AUClast (μg·h/mL) | 1.52 ± 0.47 | 1.51 ± 0.51 | 0.77 ± 0.31 | 3.12 ± 1.39 |